SCHEMBL24781572

SCHEMBL24781572

OBc1c[nH]c2ncc(Cl)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.50
CYP2C19 P33261 3/20 0.37
CYP3A4 P08684 2/20 0.37
BTK Q06187 2/20 0.36
ITK Q08881 2/20 0.36
CYP2D6 P10635 1/20 0.36
BRAF P15056 3/20 0.36
LCK P06239 3/20 0.35
KDR P35968 3/20 0.35
FLT3 P36888 3/20 0.35
MAP4K4 O95819 2/20 0.35
FYN P06241 2/20 0.35
FRK P42685 2/20 0.35
CLK2 P49760 2/20 0.35
PTK6 Q13882 2/20 0.35
NTRK3 Q16288 2/20 0.35
MINK1 Q8N4C8 2/20 0.35
SLK Q9H2G2 2/20 0.35
MAP4K5 Q9Y4K4 2/20 0.35
PRKD3 O94806 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12798698 0.83 JAK2 (0.50) JAK2CYP2C19CYP3A4CYP2D6BRAF
SCHEMBL12657249 0.77 JAK2 (0.54) JAK2CYP2C19CYP3A4BTKITK
SCHEMBL12573415 0.74 JAK2 (0.40) JAK2CYP2C19CYP3A4CYP2D6BRAF
SCHEMBL24780533 0.74 JAK2 (0.51) JAK2CYP2C19CYP3A4BTKITK
SCHEMBL18634000 0.73 JAK2 (0.42) JAK2CYP2C19CYP3A4CYP2D6BRAF
SCHEMBL29928376 0.73 JAK2 (0.54) JAK2CYP2C19CYP3A4ITKCYP2D6
SCHEMBL14883424 0.73 JAK2 (0.54) JAK2CYP2C19CYP3A4BTKITK
SCHEMBL1666074 0.73 JAK2 (0.54) JAK2CYP2C19CYP3A4ITKCYP2D6
SCHEMBL1053943 0.73 JAK2 (0.58) JAK2CYP2C19CYP3A4CYP2D6LCK
SCHEMBL15155041 0.73 GSK3B (0.56) JAK2CYP2C19CYP3A4CYP2D6LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022263801-A1 PROCESS FOR PREPARING PEXIDARTINIB JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2022-12-22 WO disclosed