SCHEMBL18634000

SCHEMBL18634000

CC(C)(C)C(C)(C)CBc1c[nH]c2ncc(Cl)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.42
CYP2C9 P11712 4/20 0.35
CYP3A4 P08684 6/20 0.34
CYP2C19 P33261 3/20 0.34
KIT P10721 3/20 0.34
LCK P06239 2/20 0.34
CSF1R P07333 2/20 0.34
PDGFRB P09619 2/20 0.34
PDGFRA P16234 2/20 0.34
FLT1 P17948 2/20 0.34
KDR P35968 2/20 0.34
FLT3 P36888 2/20 0.34
AURKB Q96GD4 2/20 0.34
PGR P06401 1/20 0.34
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CHRM1 P11229 1/20 0.34
DRD1 P21728 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12798698 0.76 JAK2 (0.50) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL21886177 0.75 GPR84 (0.46) SLC6A4MAP4K4FGFR1MAP2K1HIPK2
SCHEMBL24781572 0.73 JAK2 (0.50) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL12573415 0.71 JAK2 (0.40) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL12657250 0.71 JAK2 (0.40) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL17873349 0.70 JAK2 (0.44) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL14883424 0.68 JAK2 (0.54) JAK2CYP2C9CYP3A4CYP2C19BRAF
SCHEMBL19710201 0.67 JAK2 (0.50) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL17873389 0.66 JAK2 (0.46) JAK2CYP2C9CYP3A4CYP2C19KIT
SCHEMBL25493847 0.66 JAK2 (0.46) JAK2CYP2C9CYP3A4CYP2C19KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3141548-A1 PROCESSES AND INTERMEDIATES FOR PRODUCING AZAINDOLES Vertex Pharmaceuticals Incorporated (US) 2017-03-15 EP disclosed