SCHEMBL24784372

SCHEMBL24784372

O=C(NCc1ccccc1)c1c(O)n2ccccc2nc1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
METTL3 Q86U44 4/20 0.48
KDM4E B2RXH2 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
PKM P14618 1/20 0.47
HTT P42858 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
TP53 P04637 1/20 0.47
METTL14 Q9HCE5 2/20 0.46
TSHR P16473 1/20 0.46
SCD O00767 1/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2057951 0.86 NPC1 (0.43) NPC1KMT2AKDM4ESMN1; SMN2LMNA
SCHEMBL846337 0.78 TP53 (0.52) NPC1METTL3KDM4ESMN1; SMN2LMNA
SCHEMBL24784343 0.76 THRB (0.71) MEN1KMT2AKDM4ESMN1; SMN2LMNA
SCHEMBL24784344 0.76 THRB (0.71) MEN1KMT2AKDM4ESMN1; SMN2LMNA
SCHEMBL24784345 0.76 THRB (0.71) MEN1KMT2AKDM4ESMN1; SMN2LMNA
SCHEMBL12294853 0.75 SMN1; SMN2 (0.60) METTL3KDM4ESMN1; SMN2LMNAPKM
SCHEMBL12295463 0.74 KDM4E (0.78) NPC1KMT2AKDM4ESMN1; SMN2LMNA
SCHEMBL12294561 0.72 KDM4E (0.58) KMT2AKDM4ESMN1; SMN2LMNAPKM
SCHEMBL24784374 0.72 MAPK1 (0.60) NPC1KMT2AKDM4ESMN1; SMN2LMNA
SCHEMBL12295230 0.72 SMN1; SMN2 (0.57) KMT2AMETTL3KDM4ESMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022266473-A1 SMALL MOLECULE DISRUPTORS OF PROTEIN INTERACTIONS IN HISTONE DEACETYLASE COMPLEXES DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-12-22 WO disclosed