SCHEMBL2479401

SCHEMBL2479401

O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.57
CNR2 P34972 1/20 0.57
ALDH1A1 P00352 3/20 0.56
MGAM O43451 1/20 0.52
DPP4 P27487 1/20 0.51
PREP P48147 1/20 0.51
CHRNB2 P17787 1/20 0.50
CHRNA7 P36544 1/20 0.50
CHRNA4 P43681 1/20 0.50
KDM2B Q8NHM5 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
CA2 P00918 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
DGAT1 O75907 2/20 0.47
ACE P12821 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2479221 0.84 CNR1 (0.57) CNR1CNR2ALDH1A1DPP4CA2
SCHEMBL2474659 0.84 CNR1 (0.57) CNR1CNR2ALDH1A1DPP4CA2
SCHEMBL5740768 0.81 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2CA2L3MBTL1
SCHEMBL31313411 0.81 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2CA2L3MBTL1
SCHEMBL2476769 0.81 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2CA2L3MBTL1
SCHEMBL18586520 0.79 ACE (0.49) PREPCHRNB2CHRNA7CHRNA4ACE
SCHEMBL22811400 0.79 ACE (0.49) PREPCHRNB2CHRNA7CHRNA4ACE
SCHEMBL22798168 0.79 ACE (0.49) PREPCHRNB2CHRNA7CHRNA4ACE
SCHEMBL13229 0.78 CA2 (0.67) ALDH1A1SMN1; SMN2CA2L3MBTL1
SCHEMBL13230 0.78 CA2 (0.67) ALDH1A1SMN1; SMN2CA2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8653054-B2 2-(N-substituted piperazinyl) steroid derivatives UNIVERSITE LAVAL (CA) 2014-02-18 US disclosed
US-20110312926-A1 2-(N-Substituted Piperazinyl) Steroid Derivatives UNIVERSITE LAVAL (CA) 2011-12-22 US disclosed
EP-2373674-A1 2-(N-SUBSTITUTED PIPERAZINYL) STEROID DERIVATIVES Université Laval (CA) 2011-10-12 EP disclosed
WO-2010060215-A1 2-(N-SUBSTITUTED PIPERAZINYL) STEROID DERIVATIVES UNIVERSITé LAVAL (CA) 2010-06-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110312926-A1 2-(N-Substituted Piperazinyl) Steroid Derivatives NR5A1, HSD17B11, CYP17A1 CNR1 784/4885CNR2 1064/4885ALDH1A1 556/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.