SCHEMBL2479478

SCHEMBL2479478

COC(=O)[C@H](Cc1ccccc1)N(C(=O)OC(C)(C)C)C(=O)[C@@H](N)Cc1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
ITGA4 P13612 1/20 0.42
ITGB7 P26010 1/20 0.42
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
OPRK1 P41145 1/20 0.39
SLC7A5 Q01650 2/20 0.39
KLK5 Q9Y337 2/20 0.38
CTRB1 P17538 1/20 0.38
MC4R P32245 1/20 0.38
MC3R P41968 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LTA4H P09960 1/20 0.38
ALPI P09923 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28980532 0.85 ITGA4 (0.41) ITGA4ITGB7CTSSCTSKOPRK1
SCHEMBL11047397 0.84 SLC7A5 (0.48) ITGA4ITGB7CTSSCTSKSLC7A5
SCHEMBL17137969 0.83 ITGA4 (0.50) CA12CA7CA9CA14ITGA4
SCHEMBL13163803 0.83 ITGA4 (0.50) CA12CA7CA9CA14ITGA4
SCHEMBL7609380 0.83 ITGA4 (0.50) CA12CA7CA9CA14ITGA4
SCHEMBL2724608 0.83 ITGA4 (0.36) ITGA4ITGB7CTSKOPRK1SLC7A5
SCHEMBL1937057 0.78 ABCB1 (0.46) ITGA4ITGB7KLK5CTRB1LTA4H
SCHEMBL7269530 0.78 SLC7A5 (0.45) SLC7A5LTA4HALPIPKMPTGS1
SCHEMBL14763045 0.76 SLC7A5 (0.49) ITGA4ITGB7CTSSCTSKSLC7A5
SCHEMBL28942525 0.76 SLC7A5 (0.43) ITGA4ITGB7CTSSCTSKSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376408-A2 FLUORINATION OF ORGANIC COMPOUNDS President and Fellows of Harvard College (US) 2011-10-19 EP claimed
WO-2010059943-A2 FLUORINATION OF ORGANIC COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-05-27 WO claimed
EP-2376408-A2 FLUORINATION OF ORGANIC COMPOUNDS President and Fellows of Harvard College (US) 2011-10-19 EP disclosed
WO-2010059943-A2 FLUORINATION OF ORGANIC COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-05-27 WO disclosed