SCHEMBL2481035

SCHEMBL2481035

CNC(=O)O.O=C(N1CCCCC1)C1(c2ccccc2)CCN(C[C@@H]2C[C@@H]2c2ccc(F)c(F)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TACR3 P29371 1/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ADRA1D P25100 9/20 0.42
ADRA1A P35348 9/20 0.42
ADRA1B P35368 9/20 0.42
OPRM1 P35372 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AVPR1A P37288 1/20 0.38
NPY1R P25929 1/20 0.38
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2475976 0.84 TACR3 (0.52) HSD11B1MEN1KMT2ATACR3
SCHEMBL2476860 0.78 TACR3 (0.57) HSD11B1MEN1KMT2ATACR3ALDH1A1
SCHEMBL2481720 0.78 TACR3 (0.57) HSD11B1MEN1KMT2ATACR3ALDH1A1
SCHEMBL2474123 0.78 TACR3 (0.53) HSD11B1MEN1KMT2ATACR3
SCHEMBL2477738 0.77 TACR3 (0.53) HSD11B1TACR3
SCHEMBL2477328 0.76 TACR3 (0.53) HSD11B1MEN1KMT2ATACR3
SCHEMBL2476664 0.76 TACR3 (0.58) HSD11B1MEN1KMT2ATACR3ALDH1A1
SCHEMBL2477331 0.76 TACR3 (0.58) HSD11B1MEN1KMT2ATACR3ALDH1A1
SCHEMBL2480350 0.76 TACR3 (0.67) HSD11B1MEN1KMT2ATACR3
SCHEMBL2477401 0.76 TACR3 (0.44) HSD11B1MEN1KMT2ATACR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP claimed