SCHEMBL24813862

SCHEMBL24813862

Nc1[nH]c(=O)[nH]c(=O)c1NCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
MEN1 O00255 4/20 0.58
KMT2A Q03164 4/20 0.58
MAPT P10636 2/20 0.58
NPSR1 Q6W5P4 1/20 0.58
ALDH1A1 P00352 3/20 0.52
GAA P10253 2/20 0.52
GLA P06280 1/20 0.52
ATM Q13315 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
PNP P00491 1/20 0.47
HPGD P15428 2/20 0.46
CDC25B P30305 1/20 0.44
USP2 O75604 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4406872 0.74 ALDH1A1 (0.53) KDM4EMEN1KMT2AMAPTNPSR1
SCHEMBL7434388 0.74 KDM4E (0.67) KDM4EMEN1KMT2AMAPTNPSR1
SCHEMBL22111515 0.73 KDM4E (0.78) KDM4EMEN1KMT2AMAPTNPSR1
SCHEMBL3747115 0.72 MAPKAPK2 (0.66) KDM4EMEN1KMT2AMAPTNPSR1
SCHEMBL11678932 0.70 PNP (0.60) KDM4EMEN1KMT2AMAPTNPSR1
SCHEMBL15384307 0.69 MEN1 (0.45) MEN1KMT2ANPSR1ALDH1A1GAA
SCHEMBL16298385 0.68 ALDH1A1 (0.47) KDM4EMEN1KMT2AMAPTNPSR1
SCHEMBL18175194 0.68 TYMP (0.41) GAAPNP
SCHEMBL11760490 0.67 PNP (0.60) MEN1KMT2AMAPTALDH1A1L3MBTL1
SCHEMBL5452618 0.67 GPR84 (0.53) KDM4EMEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023122298-A1 PROTEIN STABILIZING COMPOUNDS CONTAINING USP28 AND/OR USP25 TARGETING LIGANDS Stablix, Inc. (US) 2023-06-29 WO disclosed
WO-2022272133-A2 PROTEIN STABILIZING COMPOUNDS CONTAINING USP7 LIGANDS Stablix, Inc. (US) 2022-12-29 WO disclosed