SCHEMBL2482585

SCHEMBL2482585

O=C1CNC(C(=O)c2cc(-c3ccc(F)c(Cl)c3)c(-c3cccc(Cl)c3)s2)N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
SLC9A1 P19634 2/20 0.36
CHRM1 P11229 7/20 0.33
TDP2 O95551 3/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
CHRM3 P20309 4/20 0.32
CHRM2 P08172 3/20 0.32
PGR P06401 2/20 0.32
MAPK1 P28482 3/20 0.31
LCK P06239 1/20 0.31
SRC P12931 1/20 0.31
PRKACA P17612 1/20 0.31
PRKACG P22612 1/20 0.31
PRKACB P22694 1/20 0.31
KDR P35968 1/20 0.31
FLT3 P36888 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2480657 0.88 CHRM1 (0.34) SLC9A1CHRM1TDP2HSD17B1HSD17B2
SCHEMBL2482779 0.81 HCRTR1 (0.35) BRD4TDP2HCRTR1HCRTR2PGR
SCHEMBL2479703 0.81 CA12 (0.34) SLC9A1CHRM1TDP2CHRM3CHRM2
SCHEMBL421601 0.76 MAPK14 (0.40) BRD4CREBBPSLC9A1TDP2HCRTR1
SCHEMBL10109878 0.68 MAPK14 (0.46) SLC9A1HSD17B1HSD17B2
SCHEMBL10109877 0.66 MAPK14 (0.39) SLC9A1TDP2MAPK1
SCHEMBL422068 0.65 MAPK14 (0.50) SLC9A1KDRGSK3AGSK3B
SCHEMBL424176 0.65 MAPK14 (0.37) HCRTR1HCRTR2
SCHEMBL423833 0.65 MAPK14 (0.37) HCRTR1HCRTR2
SCHEMBL424281 0.64 MAPK14 (0.42) BRD4CREBBPSLC9A1CHRM1TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376482-A1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AiCuris GmbH & Co. KG (DE) 2011-10-19 EP disclosed
WO-2010075962-A1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AICURIS GMBH & CO. KG (DE) 2010-07-08 WO disclosed