SCHEMBL2479703

SCHEMBL2479703

O=C1CNC(C(=O)c2cc(-c3cccc(Cl)c3)c(Br)s2)N1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
HSP90AA1 P07900 2/20 0.34
HSP90AB1 P08238 2/20 0.34
SLC9A1 P19634 1/20 0.34
TDP2 O95551 2/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CHRM1 P11229 8/20 0.33
CHRM3 P20309 3/20 0.33
PGR P06401 2/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
MIF P14174 1/20 0.32
CLK1 P49759 1/20 0.32
CLK2 P49760 1/20 0.32
CLK3 P49761 1/20 0.32
RORB Q92753 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2482779 0.85 HCRTR1 (0.35) HSP90AA1HSP90AB1TDP2NPC1POLB
SCHEMBL2480657 0.82 CHRM1 (0.34) HSP90AA1HSP90AB1SLC9A1TDP2NPC1
SCHEMBL2482585 0.81 BRD4 (0.39) SLC9A1TDP2CHRM1CHRM3PGR
SCHEMBL424378 0.74 RAB9A (0.43) SLC9A1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL423837 0.68 TRPM8 (0.53) NPC1RAB9ASMN1; SMN2
SCHEMBL2485716 0.64 RORB (0.39) CA12CA9SLC9A1NPC1POLB
SCHEMBL2486656 0.62 PGR (0.31) PGR
SCHEMBL10109878 0.60 MAPK14 (0.46) SLC9A1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL25356536 0.60 HSD17B10 (0.50) POLBRAB9A
SCHEMBL10109877 0.59 MAPK14 (0.39) SLC9A1TDP2NPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376482-A1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AiCuris GmbH & Co. KG (DE) 2011-10-19 EP disclosed
WO-2010075962-A1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AICURIS GMBH & CO. KG (DE) 2010-07-08 WO disclosed