SCHEMBL2483053

SCHEMBL2483053

CN(C)CC(=O)N1CCC(F)(COc2ncc(S(N)(=O)=O)cc2Cl)CC1.NS(=O)(=O)c1cnc(OCC2(F)CCNCC2)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 6/20 0.40
BCL2L1 Q07817 1/20 0.40
IRAK4 Q9NWZ3 3/20 0.35
SCN9A Q15858 3/20 0.34
SMO Q99835 1/20 0.33
LRRK2 Q5S007 1/20 0.32
TACR1 P25103 1/20 0.32
RAB9A P51151 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTR6 P50406 1/20 0.31
ADRB2 P07550 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1700098 0.95 BCL2 (0.41) BCL2BCL2L1IRAK4SCN9ASMO
SCHEMBL1959260 0.84 IRAK4 (0.38) BCL2IRAK4SCN9ALRRK2
Trifluoroacetic Acid SCHEMBL1700071 0.81 IRAK4 (0.37) IRAK4SCN9ALRRK2
SCHEMBL1700303 0.79 SCN9A (0.41) SCN9A
SCHEMBL1700322 0.79 ALDH1A1 (0.39) BCL2SCN9ALRRK2ALDH1A1
SCHEMBL1700662 0.78 CA2 (0.41) BCL2SCN9ASMO
SCHEMBL1701933 0.75 BCL2 (0.42) BCL2SCN9AALDH1A1
SCHEMBL1700545 0.75 SCN9A (0.40) BCL2SCN9A
SCHEMBL1700543 0.75 SCN9A (0.40) BCL2SCN9A
SCHEMBL1701186 0.75 SCN9A (0.40) BCL2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376197-A2 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES Abbott Laboratories (US) 2011-10-19 EP disclosed
WO-2010065824-A2 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBOTT LABORATORIES (US) 2010-06-10 WO disclosed