SCHEMBL2483240

SCHEMBL2483240

CCOC(=O)Oc1cc(-c2cccc(Cl)c2)cs1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.46
MAPT P10636 2/20 0.46
TRPM8 Q7Z2W7 1/20 0.46
RORC P51449 1/20 0.45
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
ALOX5 P09917 4/20 0.41
ABL1 P00519 1/20 0.41
DYRK3 O43781 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK2 Q92630 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
XPO1 O14980 1/20 0.40
PTGES O14684 1/20 0.39
CNR1 P21554 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
JAK2 O60674 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL426543 0.79 TRPM8 (0.53) L3MBTL1MAPTTRPM8RORCPDE4A
SCHEMBL8236043 0.77 ABL1 (0.55) L3MBTL1MAPTTRPM8RORCABL1
SCHEMBL2482550 0.77 TRPM8 (0.46) L3MBTL1MAPTTRPM8RORCPDE4A
SCHEMBL2485667 0.77 TRPM8 (0.46) L3MBTL1MAPTTRPM8PDE4APDE4B
SCHEMBL2484620 0.74 MAPT (0.46) L3MBTL1MAPTTRPM8ALOX5DYRK3
SCHEMBL28368547 0.72 MAPT (0.47) L3MBTL1MAPTTRPM8RORCPDE4A
SCHEMBL30541332 0.72 MAPT (0.47) L3MBTL1MAPTTRPM8RORCPDE4A
SCHEMBL10872998 0.71 KMT2A (0.40) L3MBTL1MAPTALOX5KDM4EALDH1A1
SCHEMBL2482717 0.71 CUL4A (0.45) L3MBTL1MAPTGABRB2KDM4EALDH1A1
SCHEMBL28369187 0.71 MAPT (0.46) L3MBTL1MAPTRORCKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376482-B1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AICURIS GMBH & CO KG (DE) 2013-03-06 EP disclosed
EP-2376482-A1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AiCuris GmbH & Co. KG (DE) 2011-10-19 EP disclosed
WO-2010075962-A1 SUBSTITUTED (THIOPHENYL-CARBONYL)IMIDAZOLIDINONES, AND USE THEREOF AICURIS GMBH & CO. KG (DE) 2010-07-08 WO disclosed