SCHEMBL2484385

SCHEMBL2484385

C=CCC1C(=O)C(=O)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.38
CASP3 P42574 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CES2 O00748 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
POLB P06746 2/20 0.36
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
HTT P42858 2/20 0.35
MITF O75030 1/20 0.35
NSD2 O96028 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTPRC P08575 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8736635 0.89 EDNRB (0.42) HTR2ACASP3CA1CA2CES2
SCHEMBL252162 0.81 HTR2A (0.52) HTR2ACA1CA2CES2ALDH1A1
SCHEMBL8546525 0.77 KDM4E (0.37) CASP3CES2KMT2AMEN1EDNRB
SCHEMBL9536703 0.72 CES2 (0.32) HTR2ACES2
SCHEMBL4552155 0.72 IDO1 (0.45) HTR2APOLBALDH1A1LMNAHTT
SCHEMBL9547888 0.72 HTR2A (0.42) HTR2ACA1CA2KMT2AMEN1
SCHEMBL11764926 0.71 EDNRB (0.47) HTR2AEDNRBEDNRAHTTCYP1A2
SCHEMBL4551141 0.70 HTR2A (0.39) HTR2ACASP3CA1CA2CES2
SCHEMBL16859501 0.70 HSD17B10 (0.55) HTR2AALDH1A1CYP1A2KDM4EHPGD
SCHEMBL5140755 0.69 CA1 (0.37) HTR2ACA1CA2CES2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364982-A1 Spiro-piperidine compounds as chemokine receptor antagonists and medicinal use thereof ONO Pharmaceutical Co., Ltd. (JP) 2011-09-14 EP disclosed
EP-1621540-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2006-02-01 EP disclosed
EP-1619193-A1 SPIROPIPERIDINE COMPOUND AND MEDICINAL USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2006-01-25 EP disclosed