SCHEMBL2484837

SCHEMBL2484837

CCOC(=O)Oc1cc(Br)c(-c2ccc(F)c(Cl)c2)o1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPA1 P27694 1/20 0.38
ALOX5 P09917 4/20 0.38
CUL4A Q13619 3/20 0.36
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
AR P10275 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSPO P30536 1/20 0.35
PTPRC P08575 1/20 0.35
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPA Q15257 1/20 0.35
TSHR P16473 2/20 0.34
KMO O15229 1/20 0.34
CASP1 P29466 1/20 0.34
ABL1 P00519 1/20 0.34
MAOB P27338 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2482175 0.84 CUL4A (0.39) CUL4AALDH1A1NPC1MAPTRAB9A
SCHEMBL2485581 0.84 ALOX5 (0.47) ALOX5CUL4AALDH1A1MAPT
SCHEMBL2484122 0.82 XPO1 (0.36) RPA1ALOX5CUL4APGRALDH1A1
SCHEMBL418485 0.81 MAOB (0.44) RPA1ALOX5ALDH1A1PTPRCPTPN2
SCHEMBL2509896 0.78 PGR (0.42) RPA1ALOX5NR3C1PGRNR3C2
SCHEMBL2510358 0.74 CNR2 (0.44) ALOX5CUL4APGRPOLB
SCHEMBL8232745 0.73 ABL1 (0.39) ALOX5CUL4ATSPOPTPRCPTPN2
SCHEMBL2486696 0.72 CUL4A (0.47) CUL4AALDH1A1TSHRMAOBPOLB
SCHEMBL2487648 0.70 ALOX5 (0.41) ALOX5ALDH1A1MAPTCHRM3
SCHEMBL15620632 0.68 ALOX5 (0.40) RPA1ALOX5ALDH1A1PTPRCPTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376479-B1 SUBSTITUTED FURANCARBOXAMIDES, AND USE THEREOF AICURIS GMBH & CO KG (DE) 2016-03-02 EP disclosed
EP-2376479-A1 SUBSTITUTED FURANCARBOXAMIDES, AND USE THEREOF AiCuris GmbH & Co. KG (DE) 2011-10-19 EP disclosed
WO-2010075957-A1 SUBSTITUTED FURANCARBOXAMIDES, AND USE THEREOF AICURIS GMBH & CO. KG (DE) 2010-07-08 WO disclosed