SCHEMBL248513

SCHEMBL248513

O=CCc1cnc2ccoc2c1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
CYP2A6 P11509 1/20 0.33
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15651507 0.79 CYP2A6 (0.46) CYP2A6
SCHEMBL10855251 0.79 NOS3 (0.36)
SCHEMBL3802865 0.79 RECQL (0.36) CYP19A1
SCHEMBL3799743 0.79 CYP19A1 (0.33) CYP19A1
SCHEMBL29935668 0.79 CYP2A6 (0.46) CYP2A6
SCHEMBL22778675 0.75 HTR1B (0.39)
SCHEMBL28063797 0.74 MEN1 (0.45)
SCHEMBL10555013 0.72 HRH3 (0.38)
SCHEMBL29950798 0.69 CHRM2 (0.56) CHRM2CHRM1CHRM3CYP2A6CYP19A1
SCHEMBL418936 0.68 DYRK1A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3810593-A1 OGA INHIBITOR COMPOUNDS Janssen Pharmaceutica NV (BE) 2021-04-28 EP disclosed
WO-2019243526-A1 OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2019-12-26 WO disclosed
EP-2588465-A1 SGC STIMULATORS Ironwood Pharmaceuticals, Inc. (US) 2013-05-08 EP disclosed
WO-2012003405-A1 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2012-01-05 WO disclosed