SCHEMBL24855201

SCHEMBL24855201

CC(C)(C)OC(=O)n1cc(C=O)c2cc(OC(F)(F)F)ccc21

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.41
KCNQ3 O43525 3/20 0.41
KCNQ2 O43526 3/20 0.41
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ELANE P08246 2/20 0.37
ACHE P22303 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
LIPE Q05469 1/20 0.35
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30844606 1.00 HTR6 (0.41) HTR6KCNQ3KCNQ2ALDH1A1KDM4E
SCHEMBL4376044 0.87 ALDH1A1 (0.48) HTR6ALDH1A1MEN1KMT2AACHE
SCHEMBL29443995 0.87 ALDH1A1 (0.48) HTR6ALDH1A1MEN1KMT2AACHE
SCHEMBL16729466 0.83 MAP2K4 (0.44) HTR6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL2461044 0.83 ALDH1A1 (0.55) HTR6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL15902182 0.83 HTR6 (0.46) HTR6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL29443980 0.83 HTR6 (0.46) HTR6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL7715925 0.81 HTR6 (0.44) HTR6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL2454469 0.81 HTR6 (0.44) HTR6ALDH1A1KDM4EMEN1KMT2A
SCHEMBL17968965 0.79 ALDH1A1 (0.61) ALDH1A1KDM4EMEN1KMT2AELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117616010-A Process for preparing (S) -2- (4-chloro-2-methoxyphenyl) -2- ((3-methoxy-5- (methylsulfonyl) phenyl) amino) -1- (1H-indol-3-yl) ketene derivatives 杨森制药公司 2024-02-27 CN disclosed
WO-2023274237-A1 PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3-METHOXY-5-(METHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES Janssen Pharmaceuticals, Inc. (US) 2023-01-05 WO disclosed