SCHEMBL24858604

SCHEMBL24858604

COC(=O)c1cc2c(Br)c(Cl)ccc2s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
HDAC1 Q13547 3/20 0.46
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC9 Q9UKV0 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
ICAM1 P05362 1/20 0.41
SELE P16581 1/20 0.41
VCAM1 P19320 1/20 0.41
CSNK2A2 P19784 2/20 0.40
CSNK2B P67870 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6331785 0.86 CCNC (0.49) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL828767 0.84 CSNK2A2 (0.44) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL30714296 0.82 RPS6KB1 (0.45) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL26110533 0.82 RPS6KB1 (0.45) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL9431710 0.82 HDAC1 (0.52) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL3822544 0.79 ICAM1 (0.41) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL829477 0.79 CCNC (0.48) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL828439 0.79 HDAC3 (0.68) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL9432038 0.78 CCNC (0.47) CCNCCDK8HDAC1HDAC3HDAC4
SCHEMBL2138333 0.78 CCNC (0.50) CCNCCDK8HDAC1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023274383-A1 KRAS G12D INHIBITOR AND USE THEREOF 上海迪诺医药科技有限公司 2023-01-05 WO disclosed
CN-115557974-A KRAS G12D inhibitor and application thereof 上海迪诺医药科技有限公司 2023-01-03 CN disclosed