SCHEMBL3822544

SCHEMBL3822544

COC(=O)c1cc2c(Br)c(C)ccc2s1.COC(=O)c1cc2c(C)c(C)ccc2s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 1/20 0.41
SELE P16581 1/20 0.41
VCAM1 P19320 1/20 0.41
CSNK2A2 P19784 2/20 0.41
CSNK2B P67870 2/20 0.41
CSNK2A1 P68400 2/20 0.41
KDR P35968 1/20 0.41
HDAC1 Q13547 2/20 0.40
PFKFB3 Q16875 2/20 0.40
PFKFB4 Q16877 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL828767 0.94 CSNK2A2 (0.44) ICAM1SELEVCAM1CSNK2A2CSNK2B
SCHEMBL829703 0.92 CSNK2A2 (0.47) ICAM1SELEVCAM1CSNK2A2CSNK2B
SCHEMBL21505451 0.81 KDM4E (0.46) ICAM1SELEVCAM1CSNK2A1HDAC1
SCHEMBL30640499 0.81 KDM4E (0.46) ICAM1SELEVCAM1CSNK2A1HDAC1
SCHEMBL26622003 0.81 PTPN2 (0.45) ICAM1SELEHDAC1HDAC3HDAC4
SCHEMBL24858604 0.79 CCNC (0.46) ICAM1SELEVCAM1CSNK2A2CSNK2B
SCHEMBL26110533 0.79 RPS6KB1 (0.45) ICAM1SELEVCAM1CSNK2A2CSNK2B
SCHEMBL9431710 0.79 HDAC1 (0.52) ICAM1SELEVCAM1CSNK2A2CSNK2B
SCHEMBL30714296 0.79 RPS6KB1 (0.45) ICAM1SELEVCAM1CSNK2A2CSNK2B
SCHEMBL829477 0.79 CCNC (0.48) ICAM1SELEVCAM1CSNK2A2CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831192-A4 BENZOTHIOPHEN-2-CARBONYLGUANIDINE DERIVATIVES, PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RES INST CHEM TECH (KR) 2009-08-19 EP disclosed
EP-1831192-A1 BENZOTHIOPHEN-2-CARBONYLGUANIDINE DERIVATIVES, PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Korea Research Institute of Chemical Technology (KR) 2007-09-12 EP disclosed
WO-2006071047-A1 BENZOTHIOPHEN-2-CARBONYLGUANIDINE DERIVATIVES, PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-07-06 WO disclosed