SCHEMBL24865205

SCHEMBL24865205

Cc1cc(N2CCC(C(F)(F)F)CC2)ccc1Nc1ccc2c(c1)OCC(=O)N2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.42
HTR2C P28335 2/20 0.42
GABRG2 P18507 3/20 0.41
GABRB3 P28472 3/20 0.41
GABRA5 P31644 3/20 0.41
DCLK1 O15075 1/20 0.37
LRRK2 Q5S007 1/20 0.37
SYK P43405 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
MAPK14 Q16539 1/20 0.36
F10 P00742 1/20 0.36
CMA1 P23946 1/20 0.35
IDH1 O75874 1/20 0.35
CYP11B2 P19099 2/20 0.35
CYP11B1 P15538 1/20 0.34
MAPK7 Q13164 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
PIK3CA P42336 2/20 0.34
HTR1D P28221 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123240 1.00 HTR1A (0.42) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865288 0.92 HTR1A (0.43) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL30336564 0.92 HTR1A (0.43) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24864870 0.91 DCLK1 (0.36) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865419 0.90 HTR1A (0.42) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL31123206 0.89 PLK1 (0.41) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865508 0.89 PLK1 (0.41) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865162 0.89 HTR1A (0.40) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL31123253 0.89 HTR1A (0.40) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865668 0.89 HTR1A (0.43) HTR1AHTR2CGABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed