SCHEMBL24865508

SCHEMBL24865508

COc1cc(N2CCC(C(F)(F)F)CC2)ccc1Nc1ccc2c(c1)OCC(=O)N2C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 3/20 0.41
TTK P33981 2/20 0.41
HTR1A P08908 4/20 0.41
HTR2C P28335 3/20 0.41
PTK2 Q05397 2/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
MAPK14 Q16539 2/20 0.39
MAPK7 Q13164 7/20 0.39
LRRK2 Q5S007 6/20 0.39
DCLK1 O15075 2/20 0.39
ALK Q9UM73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123206 1.00 PLK1 (0.41) PLK1TTKHTR1AHTR2CPTK2
SCHEMBL24865288 0.90 HTR1A (0.43) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL30336564 0.90 HTR1A (0.43) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL31123240 0.89 HTR1A (0.42) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865205 0.89 HTR1A (0.42) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865419 0.89 HTR1A (0.42) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL31123260 0.87 HTR1A (0.47) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24864940 0.87 HTR1A (0.47) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL31123189 0.87 GABRG2 (0.44) HTR1AHTR2CGABRG2GABRB3GABRA5
SCHEMBL24865342 0.87 GABRG2 (0.44) HTR1AHTR2CGABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed