SCHEMBL24865342

SCHEMBL24865342

CN1C(=O)COc2cc(Nc3ccc(N4CCC(C(F)(F)F)CC4)cc3)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
GABRA5 P31644 2/20 0.44
HTR1A P08908 3/20 0.44
HTR2C P28335 3/20 0.44
SYK P43405 2/20 0.40
IDH1 O75874 1/20 0.38
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
F10 P00742 1/20 0.37
CNR2 P34972 1/20 0.36
GRM4 Q14833 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
SLC6A4 P31645 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123189 1.00 GABRG2 (0.44) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL31123354 0.92 HTR1A (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL24865628 0.92 HTR1A (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL24864950 0.92 GABRG2 (0.44) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL24865191 0.90 CNR2 (0.36) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL24865288 0.89 HTR1A (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL30336564 0.89 HTR1A (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL24864970 0.89 GABRG2 (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL31123306 0.89 GABRG2 (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C
SCHEMBL24865336 0.89 GABRG2 (0.43) GABRG2GABRB3GABRA5HTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed