SCHEMBL2486672

SCHEMBL2486672

COc1ccccc1Cc1ncc(C(C)C(=O)O)c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.49
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
TSHR P16473 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
BRS3 P32247 1/20 0.39
CASP3 P42574 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
POLB P06746 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP2C9 P11712 1/20 0.39
HIF1A Q16665 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
PLA2G2A P14555 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1369731 0.84 HSPA5 (0.39) PTGS1PTGS2POLBL3MBTL1MAPT
SCHEMBL1369734 0.82 SLC1A5 (0.49) KMT2AMEN1HTTPOLBTP53
SCHEMBL1367547 0.81 AR (0.52) ARTSHRKMT2AMEN1PKM
SCHEMBL1369142 0.81 KDR (0.47) HTTLMNAMAPT
SCHEMBL1367422 0.78 MAPT (0.56) ARTSHRKMT2AHPGDHTT
SCHEMBL1366570 0.76 PARP1 (0.38) PTGS1PTGS2TSHR
SCHEMBL1367124 0.75 L3MBTL1 (0.38) PTGS1PTGS2TSHRPOLBL3MBTL1
SCHEMBL8473051 0.72 PTGS2 (0.64) PTGS1PTGS2KMT2AHPGDHTT
SCHEMBL7885098 0.72 PTGS2 (0.64) PTGS1PTGS2KMT2AHPGDHTT
SCHEMBL362211 0.72 PTGS2 (0.64) PTGS1PTGS2KMT2AHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2377851-A1 ISOQUINOLINE DERIVATIVE Taisho Pharmaceutical Co., Ltd. (JP) 2011-10-19 EP disclosed