SCHEMBL24869256

SCHEMBL24869256

CC(C)c1ccc2oc(-c3ccc(Cl)c(Cl)c3)nc2c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 12/20 0.70
KDM4E B2RXH2 5/20 0.70
ALDH1A1 P00352 5/20 0.70
TP53 P04637 5/20 0.70
NPC1 O15118 5/20 0.70
RAB9A P51151 5/20 0.70
HSD17B10 Q99714 3/20 0.70
MEN1 O00255 2/20 0.70
KMT2A Q03164 2/20 0.70
POLB P06746 2/20 0.58
MAOA P21397 1/20 0.56
ADRA1A P35348 1/20 0.56
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
UTRN P46939 1/20 0.54
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19806580 0.90 MAPT (0.85) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL2249285 0.89 MAOA (0.57) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL2739309 0.87 MAPT (0.76) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL19379995 0.82 RAB9A (1.00) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL23380379 0.82 KDM4E (0.78) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL2739327 0.81 MAPT (0.76) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL14275901 0.81 MAPT (0.76) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL29819651 0.81 MAPT (0.76) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL23373921 0.80 NPC1 (0.69) MAPTKDM4EALDH1A1TP53NPC1
SCHEMBL3951712 0.79 ESR1 (0.56) MAPTKDM4EALDH1A1TP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO disclosed