SCHEMBL24876146

SCHEMBL24876146

Cc1cc2[nH]c(=O)c(=O)[nH]c2c(F)c1SCl

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 18/20 0.50
GRIN2D O15399 15/20 0.50
GRIN3B O60391 15/20 0.50
GRIN2A Q12879 15/20 0.50
GRIN2B Q13224 15/20 0.50
GRIN2C Q14957 15/20 0.50
GRIN3A Q8TCU5 15/20 0.50
HSD17B10 Q99714 2/20 0.47
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24876155 0.73 GRIN1 (0.49) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL5973354 0.71 GRIN1 (0.67) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL24875986 0.68 GRIN2D (0.61) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL7786608 0.68 GRIN2D (0.65) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL7784266 0.67 GRIN2D (0.69) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL7346405 0.67 GRIN2D (1.00) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL7786519 0.67 GRIN2D (0.72) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL5973771 0.66 GRIN1 (0.68) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL121942 0.65 GRIN2D (1.00) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL463564 0.65 GRIN2D (0.70) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023280970-A1 INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2023-01-12 WO disclosed