SCHEMBL24891722

SCHEMBL24891722

CC(C)(C)OC(=O)Nc1ccc(NC(=O)C23CCC(C(=O)Nc4ccc(C5=CCN(C(=O)OC(C)(C)C)CC5)cc4)(CC2)CC3)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.63
CDK7 P50613 1/20 0.47
CDK13 Q14004 1/20 0.47
CDK12 Q9NYV4 1/20 0.47
WNT3A P56704 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
PTPN6 P29350 1/20 0.47
PDK4 Q16654 1/20 0.46
GRM1 Q13255 6/20 0.44
GRM5 P41594 5/20 0.44
HTR6 P50406 1/20 0.43
JAK1 P23458 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KIT P10721 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24891783 0.90 NAMPT (0.57) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24892373 0.89 NAMPT (0.55) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24891865 0.87 NAMPT (0.55) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24891878 0.85 NAMPT (0.51) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24891670 0.84 NAMPT (0.57) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24891972 0.84 NAMPT (0.51) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL30182359 0.84 NAMPT (0.51) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24892192 0.84 NAMPT (0.51) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL22325022 0.83 NAMPT (0.71) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24891933 0.83 NAMPT (0.55) NAMPTCDK7CDK13CDK12WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed