SCHEMBL2489989

SCHEMBL2489989

C[C@H](CC(N)=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.44
ALDH1A1 P00352 1/20 0.43
TACR1 P25103 9/20 0.41
CES2 O00748 1/20 0.41
EPHX1 P07099 3/20 0.39
ICMT O60725 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22630847 0.84 AURKA (0.59) AURKACES2EPHX1
SCHEMBL12895165 0.84 AURKA (0.59) AURKACES2EPHX1
SCHEMBL1226196 0.83 CES2 (0.45) AURKACES2
SCHEMBL1226200 0.83 CES2 (0.45) AURKACES2
SCHEMBL2692867 0.83 CES2 (0.45) AURKACES2
Hydrochloric Acid SCHEMBL6782896 0.82 ALDH1A1 (0.40) ALDH1A1TACR1CES2EPHX1ICMT
SCHEMBL7386503 0.79 CES2 (0.41) ALDH1A1TACR1CES2EPHX1GAA
SCHEMBL3143623 0.77 CES2 (0.45) AURKAALDH1A1TACR1CES2EPHX1
SCHEMBL2510406 0.77 CES2 (0.45) AURKAALDH1A1TACR1CES2EPHX1
SCHEMBL2486728 0.77 CES2 (0.45) AURKAALDH1A1TACR1CES2EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1524266-B1 Pharmaceutical composition GLAXO GROUP LTD (GB) 2007-02-28 EP claimed
EP-2117562-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING NK1 RECEPTOR ANTAGONISTS AND SODIUM CHANNEL BLOCKERS GLAXO GROUP LTD (GB) 2011-10-26 EP disclosed