SCHEMBL24900364

SCHEMBL24900364

Cc1ccc2c(c1)c(-c1nc(Cl)ncc1C(F)(F)F)cn2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.42
DYRK1A Q13627 1/20 0.35
PDK1 Q15118 1/20 0.35
CDK7 P50613 3/20 0.34
LRRK2 Q5S007 3/20 0.34
CCNH P51946 2/20 0.34
MNAT1 P51948 2/20 0.34
CDK5 Q00535 2/20 0.33
S1PR1 P21453 2/20 0.33
S1PR3 Q99500 2/20 0.33
JUN P05412 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CDK5R1 Q15078 1/20 0.33
AURKA O14965 1/20 0.33
JAK2 O60674 1/20 0.33
PAK4 O96013 1/20 0.33
ABL1 P00519 1/20 0.33
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30957591 1.00 EGFR (0.42) EGFRDYRK1APDK1CDK7LRRK2
SCHEMBL24900433 0.88 PDK1 (0.47) EGFRPDK1CDK7LRRK2CCNH
SCHEMBL30957473 0.88 PDK1 (0.47) EGFRPDK1CDK7LRRK2CCNH
SCHEMBL30221565 0.85 PDK1 (0.47) EGFRPDK1CDK7LRRK2CDK5
SCHEMBL24900656 0.85 PDK1 (0.47) EGFRPDK1CDK7LRRK2CDK5
SCHEMBL24900722 0.84 PDK1 (0.39) PDK1CDK7LRRK2CDK5CDK5R1
SCHEMBL30957512 0.84 PDK1 (0.39) PDK1CDK7LRRK2CDK5CDK5R1
SCHEMBL24900406 0.84 EGFR (0.51) EGFRPDK1CDK7CCNHMNAT1
SCHEMBL30221531 0.84 EGFR (0.51) EGFRPDK1CDK7CCNHMNAT1
SCHEMBL24900563 0.83 EGFR (0.39) EGFRDYRK1APDK1CDK7LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287783-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ACEA Therapeutics, Inc. (US) 2023-01-19 WO disclosed