SCHEMBL24900656

SCHEMBL24900656

COc1ccc2c(c1)c(-c1nc(Cl)ncc1C(F)(F)F)cn2C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.47
LCK P06239 2/20 0.45
IGF1R P08069 2/20 0.45
GSK3A P49840 2/20 0.45
GSK3B P49841 2/20 0.45
CDK7 P50613 2/20 0.45
LRRK2 Q5S007 2/20 0.45
AURKB Q96GD4 2/20 0.45
AURKA O14965 1/20 0.45
PAK4 O96013 1/20 0.45
ABL1 P00519 1/20 0.45
NTRK1 P04629 1/20 0.45
FYN P06241 1/20 0.45
CSF1R P07333 1/20 0.45
RET P07949 1/20 0.45
MET P08581 1/20 0.45
PDGFRB P09619 1/20 0.45
PIM1 P11309 1/20 0.45
FGFR1 P11362 1/20 0.45
PRKACA P17612 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30221565 1.00 PDK1 (0.47) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL17683181 0.91 ALDH1A1 (0.40) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL30957563 0.85 PDK1 (0.49) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL24900439 0.85 PDK1 (0.49) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL30957591 0.85 EGFR (0.42) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL24900433 0.85 PDK1 (0.47) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL24900364 0.85 EGFR (0.42) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL30957473 0.85 PDK1 (0.47) PDK1LCKIGF1RGSK3AGSK3B
SCHEMBL24900406 0.82 EGFR (0.51) PDK1CDK7CDK9CDK5EGFR
SCHEMBL30221531 0.82 EGFR (0.51) PDK1CDK7CDK9CDK5EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287783-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ACEA Therapeutics, Inc. (US) 2023-01-19 WO disclosed