SCHEMBL24902867

SCHEMBL24902867

CC(C(=O)OCn1ccc2c(-c3cn[nH]c3)ncnc21)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.41
TPH1 P17752 1/20 0.40
MEN1 O00255 1/20 0.38
CYP2D6 P10635 1/20 0.38
KMT2A Q03164 1/20 0.38
PTGS2 P35354 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
GRK2 P25098 2/20 0.36
ACACB O00763 2/20 0.36
ACACA Q13085 2/20 0.36
PRMT5 O14744 1/20 0.35
ROCK2 O75116 5/20 0.35
ROCK1 Q13464 5/20 0.35
GLI1 P08151 1/20 0.34
GLI2 P10070 1/20 0.34
TNK2 Q07912 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24902362 0.89 PTGS2 (0.43) PTGS1TPH1CYP2D6PTGS2TRPV1
SCHEMBL24902056 0.83 TDP1 (0.41) PTGS1TPH1PTGS2
SCHEMBL24902066 0.80 PTGS1 (0.40) PTGS1TPH1PTGS2
SCHEMBL30864377 0.78 JAK2 (0.47) TPH1MEN1CYP2D6KMT2AROCK2
SCHEMBL24902015 0.78 JAK2 (0.47) TPH1MEN1CYP2D6KMT2AROCK2
SCHEMBL24902043 0.76 JAK1 (0.49) ROCK2ROCK1
SCHEMBL30749810 0.75 SIGMAR1 (0.39) TPH1PRMT5
SCHEMBL26610240 0.72 JAK2 (0.46) TPH1ROCK2ROCK1TNK2
SCHEMBL24902073 0.71 SIGMAR1 (0.39) TPH1ACACBPRMT5ROCK2
SCHEMBL24902309 0.70 PTGS1 (0.39) PTGS1MEN1KMT2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023001045-A9 EXTERNAL ANTI-INFLAMMATORY COUPLING COMPOUND DRUG, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海椿安生物医药科技有限公司 2023-10-26 WO disclosed
WO-2023001045-A1 EXTERNAL ANTI-INFLAMMATORY COUPLING COMPOUND DRUG, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海椿安生物医药科技有限公司 2023-01-26 WO disclosed