SCHEMBL9113003

SCHEMBL9113003

[CH2]C=CC=CCc1ccc2ccoc2c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 9/20 0.43
CHRM2 P08172 2/20 0.43
CHRM1 P11229 2/20 0.43
CHRM3 P20309 2/20 0.43
CYP2A6 P11509 2/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
NFKB1 P19838 1/20 0.33
MAOA P21397 1/20 0.33
ACHE P22303 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9111859 0.78 HTR1B (0.43) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL2490953 0.74 HTR1B (0.45) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL9113881 0.74 CHRM2 (0.52) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL8040625 0.72 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL9115039 0.70 HTR1B (0.44) HTR1BCYP2A6
SCHEMBL9111536 0.69 CYP2A6 (0.40) CYP2A6MRGPRX4
SCHEMBL9110906 0.69 CHRM2 (0.49) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL507041 0.69 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL957248 0.69 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL4328740 0.69 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed