SCHEMBL24909550

SCHEMBL24909550

O=S(=O)(/C=C/c1cccnc1)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 9/20 0.69
CYP11B1 P15538 1/20 0.59
CYP11B2 P19099 1/20 0.59
ALDH1A1 P00352 1/20 0.52
NAMPT P43490 2/20 0.51
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
KDM4E B2RXH2 1/20 0.49
JUN P05412 1/20 0.49
MAPT P10636 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
GPR55 Q9Y2T6 1/20 0.49
TLR9 Q9NR96 1/20 0.48
EGFR P00533 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
VCP P55072 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27236305 1.00 NFE2L2 (0.69) NFE2L2CYP11B1CYP11B2ALDH1A1NAMPT
SCHEMBL27820280 0.83 ALDH1A1 (0.55) NFE2L2CYP11B1CYP11B2ALDH1A1NAMPT
SCHEMBL5572462 0.82 TLR9 (0.64) NFE2L2ALDH1A1TLR9EGFRKMT2A
SCHEMBL5572469 0.82 TLR9 (0.64) NFE2L2ALDH1A1TLR9EGFRKMT2A
SCHEMBL29149692 0.82 TLR9 (0.64) NFE2L2ALDH1A1TLR9EGFRKMT2A
SCHEMBL30195853 0.81 NFE2L2 (0.67) NFE2L2TLR9EGFR
SCHEMBL27328033 0.80 NFE2L2 (1.00) NFE2L2CYP11B1CYP11B2
SCHEMBL4260845 0.77 NFE2L2 (0.58) NFE2L2CYP11B1CYP11B2ALDH1A1NPC1
SCHEMBL15758243 0.77 NFE2L2 (0.62) NFE2L2CYP11B1CYP11B2ALDH1A1NPC1
SCHEMBL15758245 0.77 NFE2L2 (0.62) NFE2L2CYP11B1CYP11B2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023003882-A2 COMPOUNDS HAVING SELECTIVE INACTIVATION ACTIVITY UNIVERSITY OF NORTH CAROLINA AT WILMINGTON (US) 2023-01-26 WO disclosed