SCHEMBL249194

SCHEMBL249194

[c]1cc[nH]c2ccc3nc4ccccc4c3c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.38
ALDH1A1 P00352 5/20 0.36
MAPT P10636 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
KDM4E B2RXH2 5/20 0.34
HPGD P15428 3/20 0.34
HSD17B10 Q99714 3/20 0.34
GLA P06280 3/20 0.34
MAOA P21397 2/20 0.34
CASP1 P29466 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL356854 0.78 DYRK1A (0.35) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL8058607 0.76 DYRK1A (0.49) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL28534158 0.69 CDK4 (0.41) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL28545983 0.68 ALDH1A1 (0.41) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL23150839 0.67 RAB9A (0.45) ALDH1A1MAPTSMN1; SMN2LMNACYP3A4
SCHEMBL28537969 0.66 DYRK1A (0.37) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL28540640 0.66 DYRK1A (0.37) DYRK1ACYP3A4CDK4CCND1
SCHEMBL4503458 0.65 CDK4 (0.43) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL249195 0.65 DYRK1A (0.45) DYRK1AALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL28547076 0.64 DYRK1A (0.33) DYRK1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 101 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115350279-A anti-HER 2 combinations for the treatment of tumors 博笛生物科技有限公司 2022-11-18 CN disclosed
CN-115337402-A Combination therapeutic compositions and combination therapeutic methods for treating cancer 博笛生物科技有限公司 2022-11-15 CN disclosed
CN-115252792-A anti-EGFR combinations for the treatment of tumors 博笛生物科技有限公司 2022-11-01 CN disclosed
CN-114716555-A Compounds and compositions for targeting EGFR expressing tumors 博笛生物科技有限公司 2022-07-08 CN disclosed
CN-114671954-A Compounds and compositions targeting HER2 positive tumors 博笛生物科技有限公司 2022-06-28 CN disclosed
EP-3937939-A1 IMMUNE MODULATORY COMPOSITIONS AND METHODS FOR TREATING CANCERS Birdie Biopharmaceuticals Inc. (KY) 2022-01-19 EP disclosed
CN-113633783-A Compounds and compositions for immunotherapy 博笛生物科技有限公司 2021-11-12 CN disclosed
CN-105899539-B Compounds and compositions for immunotherapy 博笛生物科技有限公司 2021-11-09 CN disclosed
CN-112587672-A anti-PD-L1 conjugates for the treatment of tumors 博笛生物科技有限公司 2021-04-02 CN disclosed
CN-112546238-A anti-PD-L1 conjugates for the treatment of tumors 博笛生物科技有限公司 2021-03-26 CN disclosed
US-20080312206-A1 Chemical Compounds-149 ASTRAZENECA AB (SE) 2008-12-18 US disclosed
EP-1984330-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2008-10-29 EP disclosed
EP-1979332-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2008-10-15 EP disclosed
EP-1966174-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2008-09-10 EP disclosed
WO-2007091046-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-08-16 WO disclosed
WO-2007083089-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-07-26 WO disclosed
WO-2007071955-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-06-28 WO disclosed
EP-1492528-A1 ANTIDIABETIC AGENTS Warner-Lambert Company LLC (US) 2005-01-05 EP disclosed
WO-2003084535-A1 ANTIDIABETIC AGENTS WARNER-LAMBERT COMPANY LLC (US) 2003-10-16 WO disclosed
EP-1155698-A1 ORGANOBORON COMPOUNDS EXHIBITING ANTICOCCIDIAL ACTIVITIES Nitto Kasei Co., Ltd. (JP) 2001-11-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080312206-A1 Chemical Compounds-149 CSF3R, CSF1R, FLT3 DYRK1A 967/4885ALDH1A1 1081/4885MAPT 3799/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.