SCHEMBL24920872

SCHEMBL24920872

Cc1cncc(Oc2ccc(C(C)(C)c3ccc(O)cc3)cc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.46
ESR2 Q92731 4/20 0.46
CYP3A4 P08684 2/20 0.46
HPGD P15428 2/20 0.46
AR P10275 1/20 0.46
TSHR P16473 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
HTR6 P50406 1/20 0.46
ESRRG P62508 1/20 0.46
SLC6A3 Q01959 1/20 0.46
HSD17B10 Q99714 1/20 0.46
IGF1R P08069 4/20 0.41
SRC P12931 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
KDM4E B2RXH2 2/20 0.35
RAB9A P51151 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12245330 0.83 RAB9A (0.50) CYP3A4HPGDTSHRIGF1RSRC
SCHEMBL2898728 0.78 MEN1 (0.54) ESR1ESR2HPGDHSD17B10ALDH1A1
SCHEMBL4450783 0.76 ESR1 (0.73) ESR1ESR2CYP3A4HPGDAR
SCHEMBL10865719 0.76 ESR1 (0.73) ESR1ESR2CYP3A4HPGDAR
SCHEMBL4797887 0.73 IGF1R (0.43) HPGDIGF1RSRCALDH1A1MEN1
SCHEMBL2330756 0.73 TEAD4 (0.47) CYP3A4HPGDTSHRIGF1RSRC
SCHEMBL12677967 0.73 HTT (0.50) HPGDTSHRHSD17B10IGF1RSRC
SCHEMBL2904931 0.73 ESR2 (0.48) ESR1ESR2ALDH1A1MEN1KMT2A
SCHEMBL24920856 0.73 PIK3CD (0.41) IGF1RSRCKMT2AKLKB1
SCHEMBL23292685 0.72 IGF1R (0.50) CYP3A4HPGDIGF1RSRCALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed