SCHEMBL24922004

SCHEMBL24922004

COc1cnc(-c2cnon2)nc1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
PKM P14618 2/20 0.33
HSP90AA1 P07900 1/20 0.33
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
SMN1; SMN2 Q16637 3/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GRM5 P41594 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
MBOAT4 Q96T53 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921586 0.78 TNKS (0.39) NPC1RAB9AL3MBTL1PKMHSP90AA1
SCHEMBL24922005 0.77
SCHEMBL24922482 0.73 MBOAT4 (0.30) MBOAT4
SCHEMBL24922508 0.73
SCHEMBL24921559 0.73 NPC1 (0.46) NPC1RAB9APKMSMN1; SMN2ALDH1A1
SCHEMBL24921605 0.73 PDK2 (0.34) NPC1RAB9ACCR1CCR5CCR8
SCHEMBL24920882 0.73 GUCY1B2 (0.42) NPC1RAB9AL3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL24921169 0.72 CCR1 (0.67) NPC1RAB9APKMCCR1CCR5
SCHEMBL24920834 0.70 CYP1A1 (0.35) NPC1L3MBTL1CCR1CCR5CCR8
SCHEMBL24921542 0.69 FTO (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed