SCHEMBL24922503

SCHEMBL24922503

CSc1cnc(-c2nnc(C)o2)nc1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 1/20 0.44
BRD4 O60885 1/20 0.33
LRRK2 Q5S007 1/20 0.31
NOTUM Q6P988 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23576598 0.77 KDM4E (0.34) BRD4LRRK2NOTUMHPGD
SCHEMBL24922486 0.74 LRRK2 (0.36) BRD4LRRK2NOTUM
SCHEMBL24921502 0.74 NPC1 (0.40) BRD4LRRK2HPGD
SCHEMBL15599482 0.74 BRD4 (0.40) BRD4NOTUMHPGD
SCHEMBL24922483 0.70 NOTUM (0.39) NOTUMHPGD
SCHEMBL24922505 0.69
SCHEMBL24922481 0.69 ACHE (0.40) LRRK2
SCHEMBL24921486 0.68 BRD4 (0.34) BRD4LRRK2
SCHEMBL10068343 0.67 NOTUM (0.38) BRD4NOTUMHPGD
SCHEMBL24922527 0.67 L3MBTL1 (0.42) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed