SCHEMBL2492782

SCHEMBL2492782

COc1ccccc1C1(N[C@@H](Cc2ccccc2)C(=O)N(C)C)C(=O)Nc2ccc(Cl)cc21

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PYGL P06737 7/20 0.44
F11 P03951 4/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP14 P50281 1/20 0.39
CBX7 O95931 1/20 0.38
CDYL Q9Y232 1/20 0.38
KMT2A Q03164 1/20 0.38
PSMB5 P28074 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2497643 0.93 PYGL (0.39) PYGLCBX7CDYLKMT2A
SCHEMBL2498324 0.93 MMP9 (0.44) MMP9MMP8PSMB5
SCHEMBL2494983 0.91 NPC1 (0.39) PYGLF11CBX7CDYL
SCHEMBL2492829 0.90 KMT2A (0.40) PYGLCBX7CDYLKMT2A
SCHEMBL2496408 0.90 CBX7 (0.40) CBX7CDYLKMT2A
SCHEMBL2501794 0.88 CBX7 (0.39) CBX7CDYLKMT2APSMB5
SCHEMBL2498534 0.88 CBX7 (0.39) PYGLCBX7CDYLKMT2A
SCHEMBL2498800 0.88 CBX7 (0.38) PYGLCBX7CDYLKMT2APSMB5
SCHEMBL2496913 0.87 SNRNP200 (0.39) F11CBX7CDYLKMT2A
SCHEMBL2499409 0.87 CBX7 (0.38) CBX7CDYLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030499-B2 1,3-dihydro-2H-indole-2-one compound and pyrrolidine-2-one compound fused with aromatic heterocycle TAISHO PHARMACEUTICAL CO., LTD. (JP) 2011-10-04 US disclosed
US-20080318923-A1 1,3-Dihydro-2H-Indole-2-One Compound and Pyrrolidine-2-One Compound Fused With Aromatic Heterocycle TAISHO PHARMACEUTICAL CO., LTD. (JP) 2008-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080318923-A1 1,3-Dihydro-2H-Indole-2-One Compound and Pyrrolidine-2-One Compound Fused With Aromatic Heterocycle AVPR1B, AVPR1A, AVPR2 PYGL 2655/4885F11 3195/4885MMP9 999/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.