SCHEMBL2492957

SCHEMBL2492957

COc1c(NC(=O)c2ccccc2)cc(-c2ccn[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.41
TTK P33981 2/20 0.41
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
INCENP Q9NQS7 1/20 0.41
KIT P10721 1/20 0.41
SRC P12931 1/20 0.41
FLT3 P36888 1/20 0.41
NR1H4 Q96RI1 4/20 0.40
PPARG P37231 3/20 0.40
PPARA Q07869 2/20 0.40
BCAT2 O15382 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
HDAC2 Q92769 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NTRK1 P04629 1/20 0.38
ROCK2 O75116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2491307 0.90 ITK (0.42) ITKTTKAURKBINCENPKIT
SCHEMBL10134543 0.89 ITK (0.41) ITKTTKAURKBINCENPKIT
SCHEMBL6766131 0.87 HTT (0.44) ITKKITSRCFLT3ALDH1A1
SCHEMBL2489637 0.85 KIT (0.38) ITKKITSRCFLT3NR1H4
SCHEMBL1542657 0.84 CYP3A4 (0.49) ITKTTKAURKAAURKBINCENP
SCHEMBL6832471 0.76 PTGS2 (0.38) ALDH1A1KDM4EMAPK1NPC1RAB9A
SCHEMBL1542748 0.76 CYP3A4 (0.47) ITKKITSRCFLT3NR1H4
SCHEMBL6765715 0.75 ERBB2 (0.44) ALDH1A1KDM4EMAPK1NPC1RAB9A
SCHEMBL6766113 0.75 PTGS2 (0.37) ALDH1A1KDM4EMAPK1NPC1RAB9A
SCHEMBL2492954 0.75 IKBKB (0.40) BCAT2KDM4ECCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379534-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-10-26 EP claimed