SCHEMBL2492954

SCHEMBL2492954

COc1c(-c2ccccc2C(N)=O)cc(-c2ccn[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.40
CDC7 O00311 1/20 0.35
NUDT1 P36639 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
CYP3A4 P08684 3/20 0.35
CHEK1 O14757 2/20 0.34
CCNE2 O96020 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
PARP1 P09874 2/20 0.33
CSNK1A1 P48729 1/20 0.33
TYRO3 Q06418 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
BCAT2 O15382 1/20 0.33
TNFRSF1A P19438 1/20 0.32
EGFR P00533 1/20 0.32
ERBB2 P04626 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6766113 0.78 PTGS2 (0.37) CYP3A4EGFRERBB2KDM4EADORA2A
SCHEMBL6832471 0.77 PTGS2 (0.38) CYP3A4EGFRERBB2KDM4EADORA2A
SCHEMBL6765715 0.76 ERBB2 (0.44) CYP3A4EGFRERBB2KDM4EADORA2A
SCHEMBL2492957 0.75 ITK (0.41) CCNE2CCNE1CDK2BCAT2KDM4E
SCHEMBL2128919 0.74 CYP3A4 (0.52) IKBKBCDC7CYP3A4CHEK1PARP1
SCHEMBL2490531 0.73 CYP3A4 (0.54) CYP3A4TNFRSF1AEGFRERBB2ADORA2A
SCHEMBL2490533 0.73 CYP3A4 (0.54) CYP3A4TNFRSF1AEGFRERBB2ADORA2A
SCHEMBL6832451 0.70 CYP3A4 (0.52) CYP3A4TNFRSF1AERBB2
SCHEMBL2491302 0.70 RARA (0.43) CYP3A4EGFRERBB2KDM4E
SCHEMBL10134543 0.69 ITK (0.41) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379534-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-10-26 EP claimed