SCHEMBL24933494

SCHEMBL24933494

NC(=O)c1cc(-c2ccc(OCC3CNC(=O)C3)cc2)c(C(F)(F)F)[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.41
SYK P43405 6/20 0.40
PARP10 Q53GL7 5/20 0.37
PARP15 Q460N3 4/20 0.37
HSD17B1 P14061 4/20 0.35
HSD17B2 P37059 4/20 0.35
PARP2 Q9UGN5 2/20 0.35
FFAR4 Q5NUL3 2/20 0.34
CHEK2 O96017 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933356 0.86 PARP10 (0.52) PARP10PARP15PARP2FFAR4CHEK2
SCHEMBL24933633 0.85 PARP10 (0.53) PARP10PARP15PARP2FFAR4CHEK2
SCHEMBL24932946 0.84 XDH (0.42) IRAK4PARP10PARP15HSD17B1HSD17B2
SCHEMBL24933017 0.84 PRKAB2 (0.42) PARP10PARP15HSD17B1HSD17B2PARP2
SCHEMBL24933789 0.82 CHEK2 (0.42) PARP10PARP15PARP2CHEK2
SCHEMBL24933589 0.82 XDH (0.49) IRAK4PARP10PARP15HSD17B1HSD17B2
SCHEMBL24933255 0.81 CHEK2 (0.47) CHEK2
SCHEMBL24933840 0.81 PRKAB2 (0.46) PARP10PARP15HSD17B1HSD17B2FFAR4
SCHEMBL29203336 0.81 CHEK2 (0.52) IRAK4PARP10PARP15PARP2CHEK2
SCHEMBL24933256 0.81 PDK2 (0.43) HSD17B1HSD17B2FFAR4CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed