SCHEMBL24933644

SCHEMBL24933644

NC(=O)c1cc(-c2ccc(OCc3ncccc3F)cc2)c(C(F)(F)F)[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SYK P43405 8/20 0.38
DHODH Q02127 1/20 0.36
PDE10A Q9Y233 1/20 0.36
CDC7 O00311 1/20 0.35
PARP1 P09874 1/20 0.35
HSD17B1 P14061 3/20 0.35
HSD17B2 P37059 3/20 0.35
PARP15 Q460N3 2/20 0.35
PARP10 Q53GL7 2/20 0.35
MAOB P27338 1/20 0.35
PARP14 Q460N5 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
LPL P06858 1/20 0.35
LIPC P11150 1/20 0.35
LIPG Q9Y5X9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933222 0.87 PRKAB2 (0.44) SYKPDE10APARP1HSD17B1HSD17B2
SCHEMBL24933521 0.87 MAOB (0.40) DHODHPDE10AHSD17B1HSD17B2PARP15
SCHEMBL30240735 0.87 MAOB (0.40) DHODHPDE10AHSD17B1HSD17B2PARP15
SCHEMBL24933620 0.85 PARP10 (0.51) SYKDHODHPDE10APARP10
SCHEMBL30240779 0.85 PARP10 (0.51) SYKDHODHPDE10APARP10
SCHEMBL30240668 0.84 MAOB (0.39) PDE10AHSD17B1HSD17B2PARP15PARP10
SCHEMBL24933641 0.84 MAOB (0.39) PDE10AHSD17B1HSD17B2PARP15PARP10
SCHEMBL24933639 0.84 NMT1 (0.40) HSD17B1HSD17B2PARP15PARP10MAOB
SCHEMBL24933190 0.83 PRKAB2 (0.48) DHODHMAOB
SCHEMBL24933821 0.83 DHODH (0.38) DHODHPDE10APARP1HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed