SCHEMBL2493533

SCHEMBL2493533

CN1CCC[C@H]1CCN(CC1CCCCC1)S(=O)(=O)c1ccc2c(c1)CNCC2

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.48
HTR2B P41595 3/20 0.48
PNMT P11086 6/20 0.42
HTR2A P28223 7/20 0.40
HTR7 P34969 7/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
BCHE P06276 2/20 0.37
NMT1 P30419 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1241177 0.77 PNMT (0.53) HTR2CHTR2BPNMTHTR2AADRA2A
SCHEMBL2403756 0.77 PNMT (0.53) HTR2CHTR2BPNMTHTR2AADRA2A
Hydrochloric Acid SCHEMBL2405913 0.76 PNMT (0.52) HTR2CHTR2BPNMTHTR2AADRA2A
Hydrochloric Acid SCHEMBL1242900 0.76 PNMT (0.52) HTR2CHTR2BPNMTHTR2AADRA2A
SCHEMBL5628447 0.72 PNMT (0.52) HTR2CHTR2BPNMTHTR2AADRA2A
SCHEMBL1077845 0.67 HTR2C (0.82) HTR2CHTR2BPNMTADRA2AADRA2B
SCHEMBL2400927 0.66 HRH3 (0.46) HTR7
SCHEMBL1241268 0.66 HRH3 (0.46) HTR7
Hydrochloric Acid SCHEMBL11738740 0.66 HTR2C (0.80) HTR2CHTR2BPNMTADRA2AADRA2B
Water SCHEMBL16161850 0.66 HRH3 (0.46) HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2542530-A2 PROCESS FOR THE PREPARATION OF 2-(CYCLOHEXYLMETHYL)-N-{2- [(2S)-1-METHYLPYRROLIDIN-2-YL]ETHYL}-1, 2, 3, 4- TETRAHYDROISOQUINOLINE-7-SULFONAMIDE SANOFI (FR) 2013-01-09 EP disclosed
WO-2011109675-A2 PROCESS FOR THE PREPARATION OF 2-(CYCLOHEXYLMETHYL)-N-{2- [(2S)-1-METHYLPYRROLIDIN-2-YL]ETHYL}-1, 2, 3, 4- TETRAHYDROISOQUINOLINE-7-SULFONAMIDE SANOFI (FR) 2011-09-09 WO disclosed