SCHEMBL2493747

SCHEMBL2493747

C#Cc1ccc(C(=C)c2ccc[nH]2)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.32
ATM Q13315 1/20 0.31
HAO1 Q9UJM8 1/20 0.31
GAA P10253 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA7 P43166 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9533233 0.77 RAB9A (0.46) RAB9ASMN1; SMN2MEN1KMT2ACYP2D6
SCHEMBL5067712 0.74 TSHR (0.43) RAB9ASMN1; SMN2NPC1MEN1KMT2A
SCHEMBL28302892 0.74 MEN1 (0.48) MEN1KMT2AHSD17B10
Phenylacetylene SCHEMBL27678817 0.67 MEN1 (0.45) MEN1KMT2AHSD17B10TSHR
SCHEMBL859852 0.67 HDAC8 (0.58) MEN1KMT2AHSD17B10CYP2D6CA12
SCHEMBL13656487 0.66 TSHR (0.43) RAB9ASMN1; SMN2NPC1MEN1KMT2A
SCHEMBL23950227 0.65 HDAC8 (0.39) CA12CA1CA2CA9
SCHEMBL13784878 0.65 CA12 (0.40) CA12CA1CA2CA9
SCHEMBL9536998 0.64 CES2 (0.45) RAB9ANPC1MEN1KMT2A
SCHEMBL3838955 0.64 SRD5A2 (0.48) CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030482-B2 3-beta-tetrahydropyranyloxy-22-[4-(4,4-difluoro-1,3,5,7-tetramethyl-4-bora-3a,4a-diaza-s-indacene-8-yl)butyroxy]-23-bisnorchol-5-ene, used in fluorescence spectroscopy for monitoring exchange, distribution and trafficking of cholesterol between living cells and lipid domains in membranes RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2011-10-04 US disclosed
US-20080177059-A1 FREE CHOLESTEROL ANALOGS BEARING A BORON DIPYRROMETHENE DIFLUORO (BODIPY) FLUOROPHORE IN THE SIDE CHAIN AND METHOD OF PREPARATION AND USE THEREOF RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK 2008-07-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080177059-A1 FREE CHOLESTEROL ANALOGS BEARING A BORON DIPYRROMETHENE DIFLUORO (BODIPY) FLUOROPHORE IN THE SIDE CHAIN AND METHOD OF PREPARATION AND USE THEREOF NPC1L1, CETP, NPC1 RAB9A 747/4885SMN1; SMN2 4159/4885NPC1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.