SCHEMBL24944905

SCHEMBL24944905

Brc1ccc(CSc2nccn2-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 1.00
CYP2C9 P11712 7/20 1.00
L3MBTL1 Q9Y468 6/20 1.00
CYP1A2 P05177 6/20 1.00
CYP2D6 P10635 6/20 1.00
CYP2C19 P33261 6/20 1.00
ALOX15B O15296 3/20 1.00
GAA P10253 2/20 0.77
ALDH1A1 P00352 5/20 0.63
SMN1; SMN2 Q16637 4/20 0.61
RAB9A P51151 3/20 0.61
NPC1 O15118 1/20 0.61
TERT O14746 1/20 0.51
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ALOX12 P18054 1/20 0.49
LMNA P02545 3/20 0.48
OPRK1 P41145 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24944906 0.87 CYP1A2 (1.00) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24943934 0.86 L3MBTL1 (0.77) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24944902 0.83 L3MBTL1 (1.00) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24945027 0.83 CYP1A2 (0.78) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24945136 0.78 L3MBTL1 (0.65) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24943937 0.78 ALDH1A1 (1.00) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL6765169 0.77 CYP1A2 (0.67) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24945138 0.76 CYP1A2 (1.00) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL24945135 0.74 L3MBTL1 (1.00) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6
SCHEMBL9377266 0.74 L3MBTL1 (0.59) CYP3A4CYP2C9L3MBTL1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023009347-A1 COMPOUNDS FOR MODULATING EPITHELIAL 15-(S)-LIPOXYGENASE-2 AND METHODS OF USE FOR SAME THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-02 WO disclosed