SCHEMBL2494619

SCHEMBL2494619

O=C(Nc1ccccn1)c1cncc(N2CCN(S(=O)(=O)c3ccsc3)CC2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.47
RAB9A P51151 6/20 0.47
NPC1 O15118 4/20 0.47
TSHR P16473 4/20 0.45
HTT P42858 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 2/20 0.44
POLB P06746 1/20 0.43
LMNA P02545 4/20 0.42
F13A1 P00488 1/20 0.42
TGM2 P21980 1/20 0.42
TGM1 P22735 1/20 0.42
GSK3B P49841 1/20 0.42
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
CRHBP P24387 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10256309 0.89 RAB9A (0.55) GRM5RAB9ANPC1TSHRHTT
SCHEMBL10255275 0.86 GRM5 (0.50) GRM5RAB9ANPC1TSHRHTT
SCHEMBL2497238 0.85 LMNA (0.60) GRM5RAB9ANPC1TSHRL3MBTL1
SCHEMBL616029 0.84 GRM5 (0.51) GRM5RAB9ANPC1TSHRHTT
SCHEMBL10255288 0.83 GRM5 (0.57) GRM5RAB9ANPC1TSHRHTT
SCHEMBL10255410 0.80 GRM5 (0.51) GRM5RAB9ANPC1TSHRHTT
SCHEMBL10255402 0.80 KDM4E (0.58) GRM5POLBALDH1A1KDM4EKMT2A
SCHEMBL10257099 0.79 GRM5 (0.50) GRM5RAB9ATSHRGAALMNA
SCHEMBL10255321 0.76 GRM5 (0.56) GRM5RAB9ANPC1TSHRHTT
SCHEMBL14822725 0.75 GRM5 (0.55) GRM5TSHRHTTL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2370424-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2011-10-05 EP disclosed