SCHEMBL24947192

SCHEMBL24947192

CC(C)(C)OC(=O)N1CCC(c2cccc(O)c2O)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 8/20 0.51
KDM4E B2RXH2 2/20 0.50
MAPT P10636 1/20 0.50
THRB P10828 1/20 0.50
NAMPT P43490 1/20 0.48
TERT O14746 1/20 0.47
STS P08842 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
PTPN6 P29350 1/20 0.47
PKM P14618 1/20 0.46
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31321884 1.00 GPR119 (0.51) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL1613087 0.89 GPR119 (0.56) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL921685 0.87 GPR119 (0.50) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL30431475 0.87 GPR119 (0.49) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL24793975 0.87 GPR119 (0.49) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL24793973 0.87 GPR119 (0.49) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL29709671 0.87 GPR119 (0.49) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL25003975 0.86 GPR119 (0.48) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL22697070 0.86 TERT (0.39) GPR119KDM4EMAPTTHRBNAMPT
SCHEMBL3436365 0.82 GPR119 (0.58) GPR119KDM4EMAPTTHRBNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117222631-A Phenyl- [1,3] dioxolo [4,5-C ] pyridinyl-phenyl-, phenyl- [1,3] dioxolo [4,5-C ] pyridinyl-heteroaryl-or phenyl- [1,3] dioxolo [4,5-C ] pyridinyl-piperidinyl-methyl-oxetanylmethyl-1H-benzo [ D ] imidazole-carboxylic acid derivatives and methods of use thereof 诚益生物(美国)公司 2023-12-12 CN disclosed
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2023000834-A1 BENZIMIDAZOLE OR AZABENZIMIDAZOLE-6-CARBOXYLIC ACID COMPOUND AND USE THEREOF 广州必贝特医药股份有限公司 2023-01-26 WO disclosed
WO-2023000834-A1 BENZIMIDAZOLE OR AZABENZIMIDAZOLE-6-CARBOXYLIC ACID COMPOUND AND USE THEREOF 广州必贝特医药股份有限公司 2023-01-26 WO disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed
US-20220348564-A1 PHENYL-[1,3]DIOXOLO[4,5-C]PYRIDINYL-PHENYL-, PHENYL-[1,3]DIOXOLO[4,5-C]PYRIDINYL-HETEROARYL-, OR PHENYL-(1,3)DIOXO[4,5-C]PYRIDINYL-PIPERIDINYL-METHYL-OXETANYLMETHYL-1H-BENZO[D]IMIDAZOLE-CARBOXYLIC ACID DERIVATIVES AND METHODS OF USING SAME ECCOGENE (SHANGHAI) CO., LTD. (CN) 2022-11-03 US disclosed
CN-113480534-B Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药股份有限公司 2022-05-13 CN disclosed
CN-113480534-A Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药技术有限公司 2021-10-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220348564-A1 PHENYL-[1,3]DIOXOLO[4,5-C]PYRIDINYL-PHENYL-, PHENYL-[1,3]DIOXOLO[4,5-C]PYRIDINYL-HETEROARYL-, OR PHENYL-(1,3)DIOXO[4,5-C]PYRIDINYL-PIPERIDINYL-METHYL-OXETANYLMETHYL-1H-BENZO[D]IMIDAZOLE-CARBOXYLIC ACID DERIVATIVES AND METHODS OF USING SAME GLP1R, GIPR, SLC5A1 GPR119 6/4885KDM4E 2093/4885MAPT 184/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.