SCHEMBL2495417

SCHEMBL2495417

CCCCCc1ccc[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.46
LIPG Q9Y5X9 1/20 0.44
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
BID P55957 3/20 0.41
MCL1 Q07820 3/20 0.41
BCL2L1 Q07817 2/20 0.41
BAK1 Q16611 2/20 0.41
KAT8 Q9H7Z6 2/20 0.41
PPARA Q07869 2/20 0.41
PPARG P37231 1/20 0.41
EP300 Q09472 1/20 0.41
KAT2A Q92830 1/20 0.41
KAT2B Q92831 1/20 0.41
KAT5 Q92993 1/20 0.41
SAE1 Q9UBE0 1/20 0.41
ALOX5 P09917 1/20 0.40
PTGS2 P35354 1/20 0.40
DAO P14920 1/20 0.39
AURKA O14965 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27397512 0.98 GPR84 (0.49) GPR84LIPGNR1H2NR1H3BID
SCHEMBL28243243 0.98 GPR84 (0.49) GPR84LIPGNR1H2NR1H3BID
SCHEMBL5166986 0.98 GPR84 (0.49) GPR84LIPGNR1H2NR1H3BID
SCHEMBL14974903 0.98 GPR84 (0.49) GPR84LIPGNR1H2NR1H3BID
SCHEMBL10767574 0.98 GPR84 (0.49) GPR84LIPGNR1H2NR1H3BID
SCHEMBL10764266 0.98 GPR84 (0.49) GPR84LIPGNR1H2NR1H3BID
SCHEMBL10692239 0.94 DAO (0.41) GPR84LIPGNR1H2NR1H3BID
SCHEMBL9234355 0.88 DAO (0.45) GPR84LIPGNR1H2NR1H3BID
SCHEMBL174911 0.86 KDM4E (0.44) GPR84MCL1DAOAURKAAURKB
SCHEMBL28003330 0.81 BID (0.44) GPR84BIDMCL1BCL2L1BAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 57 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106905230-A A kind of preparation method of aryl pyridinones compound 周晓芳 2017-06-30 CN claimed
CN-104923165-B A kind of derivant based on aryl pyridones molecular skeleton and its application in preparing hydrargyrum trapping agent 广东工业大学 2017-03-01 CN claimed
CN-104923165-A Derivative based on aromatic pyridone molecular skeleton, and application thereof in preparing mercury capturing agent UNIV GUANGDONG TECHNOLOGY 2015-09-23 CN claimed
CN-102786467-A N-substitutional aryl pyridine ketone compound as well as preparation method and application of N-substitutional aryl pyridine ketone compound ZHEJIANG ACADEMY MEDICAL SCI 2012-11-21 CN claimed
CN-113897631-B Method for electrochemical synthesis of pyridin-2-one derivatives 昆明学院 2023-05-09 CN disclosed
CN-113897631-A Method for electrochemically synthesizing pyridine-2-one derivatives 昆明学院 2022-01-07 CN disclosed
CN-110256405-A 5- alkyl-N- substituted aryl Pyridione derivatives and its preparation method and application 四川国康药业有限公司 2019-09-20 CN disclosed
CN-106397408-B 5- methyl -2 (1H) Pyridione derivatives and its preparation method and application 四川大学 2019-04-02 CN disclosed
CN-105793251-B Heteroaryl pyridines ketone with electrophilic functionality and azepine-pyridinone compounds 豪夫迈·罗氏有限公司 2018-10-12 CN disclosed
CN-107922431-A HPK1 inhibitors and methods of use thereof 大学健康网络 2018-04-17 CN disclosed
CN-105175326-B 5 methyl 2 (1H) Pyridione derivatives and its production and use 四川国康药业有限公司 2018-02-27 CN disclosed
CN-105085383-B 5 methyl 2 (1H) Pyridione derivatives and its production and use 四川大学 2017-09-01 CN disclosed
US-4866078-A Phenyl pyridones and insectidal use thereof IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-09-12 US disclosed
EP-0259048-A2 Chemical compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-03-09 EP disclosed
US-4725607-A MITICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-02-16 US disclosed
US-4725607-A MITICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-02-16 US disclosed
EP-0216541-A1 Aryl pyridones IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-04-01 EP disclosed
EP-0216541-A1 Aryl pyridones IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-04-01 EP disclosed
CN-86106734-A ARYL PYRIDONES 1987-04-01 CN disclosed
CN-86106734-A ARYL PYRIDONES 1987-04-01 CN disclosed