SCHEMBL2495486

SCHEMBL2495486

O=C(Nc1cnc(Nc2cccnc2)nc1)c1cc(Nc2ccc3ccccc3n2)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 11/20 0.51
CYP11B2 P19099 1/20 0.48
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
BTK Q06187 3/20 0.47
HTT P42858 1/20 0.45
BLK P51451 3/20 0.44
SGMS2 Q8NHU3 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14286493 0.92 RAB9A (0.51) RAB9ANPC1BTKHTTBLK
SCHEMBL14311107 0.89 BTK (0.56) BTKBLK
SCHEMBL5994609 0.79 CYP11B2 (0.56) CSF1RCYP11B2SGMS2
SCHEMBL2494628 0.79 KDR (0.42) RAB9ANPC1BTK
SCHEMBL5997052 0.77 CSF1R (0.64) CSF1RCYP11B2RAB9ANPC1SGMS2
SCHEMBL5814463 0.76 CSF1R (0.70) CSF1RCYP11B2
SCHEMBL2492453 0.75 NPC1 (0.54) RAB9ANPC1
SCHEMBL2494867 0.74 CSF1R (0.70) CSF1RBTK
SCHEMBL2491995 0.73 CSF1R (0.84) CSF1RBTKBLK
SCHEMBL19477453 0.73 CSF1R (0.60) CSF1RCYP11B2NPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030487-B2 2-amino—5-substituted pyrimidine inhibitors TARGEGEN, INC. (US) 2011-10-04 US disclosed
US-8030487-B2 2-amino—5-substituted pyrimidine inhibitors TARGEGEN, INC. (US) 2011-10-04 US disclosed
US-8030487-B2 2-amino—5-substituted pyrimidine inhibitors TARGEGEN, INC. (US) 2011-10-04 US disclosed
US-20080027070-A1 2-AMINO--5-SUBSTITUTED PYRIMIDINE INHIBITORS TARGEGEN, INC. (US) 2008-01-31 US disclosed
US-20080027070-A1 2-AMINO--5-SUBSTITUTED PYRIMIDINE INHIBITORS TARGEGEN, INC. (US) 2008-01-31 US disclosed
US-20080027070-A1 2-AMINO--5-SUBSTITUTED PYRIMIDINE INHIBITORS TARGEGEN, INC. (US) 2008-01-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080027070-A1 2-AMINO--5-SUBSTITUTED PYRIMIDINE INHIBITORS KDR, FLT4, FLT1 CSF1R 575/4885CYP11B2 3715/4885RAB9A 3189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.