SCHEMBL24955686

SCHEMBL24955686

Cn1cc(-c2ccccc2)nc1C#Cc1nc(N2C[C@H]3COC[C@H]3C2)c2ncn(C)c2n1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 8/20 0.38
ADORA1 P30542 2/20 0.35
MAP3K12 Q12852 1/20 0.33
PIK3CA P42336 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
TSPO P30536 1/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
MAPK14 Q16539 1/20 0.30
LRRK2 Q5S007 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30202390 1.00 PDE10A (0.38) PDE10AADORA1MAP3K12PIK3CAADORA3
SCHEMBL24955640 0.86 PIK3CA (0.47) PDE10AADORA1PIK3CALRRK2
SCHEMBL31106972 0.85 DGAT1 (0.38)
SCHEMBL24955726 0.85 DGAT1 (0.38)
SCHEMBL24956765 0.84 LRRK2 (0.34) ADORA1MAP3K12PIK3CAADORA3TSPO
SCHEMBL30202293 0.84 LRRK2 (0.34) ADORA1MAP3K12PIK3CAADORA3TSPO
SCHEMBL30203054 0.84 CNR2 (0.38) PDE10AADORA1MAP3K12PIK3CA
SCHEMBL30202075 0.83 PDE10A (0.37) PDE10APIK3CACHRNB2CHRNA7CHRNA4
SCHEMBL30202168 0.81 MTOR (0.49) PDE10APIK3CA
SCHEMBL30202248 0.81 MTOR (0.49) PDE10APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023007185-A1 IMIDAZOLE ORGANIC COMPOUNDS AND THEIR USE AGAINST INFLAMMATORY BOWEL DISEASE Benevolentai Cambridge Limited (GB) 2023-02-02 WO disclosed