SCHEMBL24959817

SCHEMBL24959817

O=C(Cl)c1ccc(C(F)(F)F)cc1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.50
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
AVPR2 P30518 1/20 0.44
GPR27 Q9NS67 1/20 0.44
TAS2R14 Q9NYV8 1/20 0.43
CFTR P13569 1/20 0.42
USP2 O75604 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CES1 P23141 1/20 0.39
SLC6A9 P48067 1/20 0.39
PTPN1 P18031 3/20 0.39
PTPN6 P29350 1/20 0.39
PTPN11 Q06124 1/20 0.39
MAPT P10636 1/20 0.39
XBP1 P17861 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL475119 0.85 CES2 (0.50) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL422332 0.83 ALDH1A1 (0.62) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30519391 0.81 CES2 (0.50) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2477164 0.81 CES2 (0.50) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3023134 0.81 CES2 (0.53) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL496324 0.79 GAA (0.54) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30518051 0.79 CES2 (0.72) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL937022 0.79 CES2 (0.72) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL11143987 0.79 CES2 (0.52) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL27966822 0.79 CES2 (0.52) CES2KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116874441-A Flexible aryl formamide derivative containing 1,2, 4-oxadiazole as well as preparation method and application thereof 贵州大学 2023-10-13 CN disclosed
WO-2023288253-A1 SMALL MOLECULES INHIBITORS OF CYCLIC GMP-AMP SYNTHASE (CGAS) THE SCRIPPS RESEARCH INSTITUTE (US) 2023-01-19 WO disclosed