SCHEMBL2496022

SCHEMBL2496022

CC(C#N)c1cccc2[nH]cnc12

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.41
BRD4 O60885 2/20 0.38
DRD4 P21917 3/20 0.33
DRD3 P35462 3/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
DRD2 P14416 2/20 0.33
EGFR P00533 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PRNP P04156 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2611049 0.81 PARP1 (0.46) PARP1BRD4DRD4DRD3DRD2
SCHEMBL24351926 0.78 PARP1 (0.44) PARP1BRD4DRD4DRD3DRD2
SCHEMBL7856459 0.78 PARP1 (0.47) PARP1BRD4DRD4DRD3DRD2
SCHEMBL18713659 0.75 TSHR (0.42) PARP1BRD4DRD4DRD3DRD2
SCHEMBL2127998 0.75 PARP1 (0.41) PARP1BRD4DRD4DRD3DRD2
SCHEMBL2127994 0.74 HTR2A (0.47) PARP1BRD4DRD4DRD3DRD2
SCHEMBL2496016 0.74 PARP1 (0.35) PARP1SMN1; SMN2
SCHEMBL20032408 0.73 PARP1 (0.42) PARP1BRD4DRD4DRD3DRD2
SCHEMBL2497545 0.73 PARP1 (0.50) PARP1BRD4
SCHEMBL2820806 0.72 PARP1 (0.56) PARP1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373628-A1 NOVEL COMPOUNDS Glaxo Group Limited (GB) 2011-10-12 EP disclosed
WO-2010070021-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2010-06-24 WO disclosed