SCHEMBL2496039

SCHEMBL2496039

COCCc1ncc[nH]1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593822 0.89 TERT (0.42)
SCHEMBL593619 0.89 TERT (0.42)
SCHEMBL27831718 0.89 TERT (0.42)
SCHEMBL1899700 0.88 TBXAS1 (0.49)
SCHEMBL9216061 0.83 TERT (0.50)
SCHEMBL8368761 0.80 TERT (0.44)
SCHEMBL285224 0.79 TERT (0.59)
SCHEMBL7235494 0.79
SCHEMBL7358906 0.79
SCHEMBL27748791 0.79 TERT (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2158199-A1 PIPERIDINE COMPOUNDS AND USES THEREOF AstraZeneca AB (SE) 2010-03-03 EP claimed
WO-2008152418-A1 PIPERIDINE COMPOUNDS AND USES THEREOF ASTRAZENECA AB (SE) 2008-12-18 WO claimed
WO-2023086383-A1 SELECT KRAS G12C INHIBITORS AND USES THEREOF 1200 PHARMA LLC (US) 2023-05-19 WO disclosed
WO-2022266015-A1 FUSED HETEROARYL COMPOUNDS USEFUL AS ANTICANCER AGENTS KUMQUAT BIOSCIENCES INC. (US) 2022-12-22 WO disclosed
US-11358957-B2 Microbiocidal oxadiazole derivatives SYNGENTA PARTICIPATIONS AG (CH) 2022-06-14 US disclosed
US-20200277287-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2020-09-03 US disclosed
US-20140205537-A1 LRRK2 INHIBITORS ZENOBIA THERAPEUTICS, INC. (US) 2014-07-24 US disclosed
WO-2012178015-A2 LRRK2 INHIBITORS ZENOBIA THERAPEUTICS, INC. (US) 2012-12-27 WO disclosed
US-8030339-B2 Imidazole derivatives for the treatment of anxiety and related diseases NEUROSEARCH A/S (DK) 2011-10-04 US disclosed
CN-1812789-B Sulfonamide substituted imidazoquinolines 3M INNOVATION CO LTD 2010-07-14 CN disclosed
EP-2158199-A1 PIPERIDINE COMPOUNDS AND USES THEREOF AstraZeneca AB (SE) 2010-03-03 EP disclosed
EP-0455909-A2 5-[1-(Imidazol)methyl]-3,3-disubstituted-2(3H) furanone derivatives MARION MERRELL DOW INC. (US) 1991-11-13 EP disclosed
US-5039691-A Anticholinergic agents MARION MERRELL DOW INC. (US) 1991-08-13 US disclosed
US-4307105-A FUNGICIDES AND BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1981-12-22 US disclosed
US-4307105-A FUNGICIDES AND BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1981-12-22 US disclosed
US-4260616-A FUNGICIDES, BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1981-04-07 US disclosed
US-4260616-A FUNGICIDES, BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1981-04-07 US disclosed
US-4248881-A BACTERICIDES, FUNGICIDES E. R. SQUIBB & SONS, INC. (US) 1981-02-03 US disclosed
US-4234589-A FUNGICIDES; BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1980-11-18 US disclosed
US-4234589-A FUNGICIDES; BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1980-11-18 US disclosed